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Name Synonyms FDA Status Company Target Type Therapy Type Approved
For
ABT-288 Alzheimer's Disease (Discontinued) AbbVie Cholinergic System, Other Neurotransmitters Small Molecule
Besipirdine HCl HP 749 Alzheimer's Disease (Discontinued) Aventis Pharmaceuticals, Inc. (was Hoechst) Other Neurotransmitters Small Molecule
BI 409306 SUB 166499 Alzheimer's Disease (Discontinued), Schizophrenia (Phase 2) Boehringer Ingelheim Other Neurotransmitters, Other Small Molecule
CX516 Ampalex Alzheimer's Disease (Discontinued) Cortex Pharmaceuticals, Inc. Other Neurotransmitters Small Molecule None
Dimebon Dimebolin,
Latrepirdine,
Pf-01913539
Alzheimer's Disease (Discontinued), Huntington's Disease (Discontinued) Medivation, Inc. Other Neurotransmitters, Unknown Small Molecule Anti-histamine use in Russia
GSK239512 Alzheimer's Disease (Discontinued) GlaxoSmithKline (GSK) Cholinergic System, Other Neurotransmitters Small Molecule
Iclepertin BI 425809 Alzheimer's Disease (Discontinued), Schizophrenia (Phase 3) Boehringer Ingelheim Other Neurotransmitters Small Molecule
Idalopirdine Lu AE58054,
SGS 518
Alzheimer's Disease (Discontinued), Schizophrenia (Inactive) Lundbeck, Otsuka Pharmaceutical Co., Ltd. Other Neurotransmitters Small Molecule
Intepirdine RVT-101,
SB 742457 ,
GSK 742457
Alzheimer's Disease (Discontinued), Dementia with Lewy Bodies (Discontinued) Axovant Sciences Ltd. Other Neurotransmitters Small Molecule
Neramexane MRZ 2/579 Alzheimer's Disease (Discontinued) Forest Laboratories, Inc., Merck Other Neurotransmitters Small Molecule None
NS2330 Tesofensine Alzheimer's Disease (Discontinued) NeuroSearch A/S Other Neurotransmitters Small Molecule
PF-05212377 PF-5212377,
WYE-103760,
SAM-760
Alzheimer's Disease (Discontinued) Pfizer Other Neurotransmitters Small Molecule
PXT864 PXT00864 Alzheimer's Disease (Discontinued) Pharnext Other Neurotransmitters Combination, Small Molecule
S 38093 Alzheimer's Disease (Discontinued) Servier Cholinergic System, Other Neurotransmitters Small Molecule
S47445 CX1632 Alzheimer's Disease (Discontinued) Cortex Pharmaceuticals, Inc., Servier Other Neurotransmitters Small Molecule
SB 202026 Memric Alzheimer's Disease (Discontinued) Other Neurotransmitters Small Molecule
Sembragiline RO4602522,
RG1577
Alzheimer's Disease (Discontinued) Evotech AG Other Neurotransmitters, Other Small Molecule
SGS-742 CGP-36742,
DVD-742
Alzheimer's Disease (Discontinued) Novartis Pharmaceuticals Corporation, Saegis Pharmaceuticals, Inc. Other Neurotransmitters Small Molecule
Suritozole MD 26479 Alzheimer's Disease (Discontinued) Aventis Pharmaceuticals, Inc. (was Hoechst) Other Neurotransmitters Small Molecule
Troriluzole BHV-4157, trigriluzole, FC-4157 Alzheimer's Disease (Discontinued) Biohaven Pharmaceuticals Other Neurotransmitters Other
Xaliproden SR 57746A Alzheimer's Disease (Discontinued) Sanofi Other Neurotransmitters, Other Small Molecule